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Tocris Bioscience™ SGC GAK 1
Description
SGC GAK 1 is a high affinity cyclin G associated kinase (GAK) inhibitor (Kd = 1.9 nM). Exhibits >30-fold selectivity for GAK over a panel of other kinases. Inhibits GAK in live cell assays (IC50 = 110 nM).
Specifications
Specifications
| Chemical Name or Material | 6-Bromo-N-(3,4,5-trimethoxyphenyl)-4-quinolinamine |
| CAS | 2226517-76-4 |
| Quantity | 5 mg |
| Molecular Formula | C18H17BrN2O3 |
| Purity | 99% |