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Tocris Bioscience™ Perlapine
Description
Perlapine is a potent muscarinic DREADD agonist (pEC50 values are 8.38, 8.08 and 7.27 for hM1Dq, hM3Dq and hM4Di in vitro, respectively). Exhibits >10,000-fold selectivity for hM3Dq over hM3 receptors.
Specifications
Specifications
| Chemical Name or Material | 6-(4-Methyl-1-piperazinyl)-11 H-dibenz[b,e]azepine |
| CAS | 11-3-1977 |
| Quantity | 50 mg |
| Target | DREADD Activators |
| Molecular Formula | C19H21N3 |
| Formula Weight | 291.39 |
| Purity | 99% |