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Tocris™ TCS PIM-1 4a

Selective, ATP-competitive Pim kinase inhibitor

$140.08 - $589.90

Specifications

Product Type TCS PIM-1 4a
Inhibitors TCS PIM-1 4a
Molecular Weight 273.23
Purity >98
View More Specs

 Disclaimers

For Research Use Only

Products
Catalog Number Mfr. No. Quantity Price Quantity    

371410R

 
tocris™
3714/10
10mg Each for $140.08

371450R

 
tocris™
3714/50
50mg Each for $589.90
Description & Specifications

Specifications

Product Type TCS PIM-1 4a
Inhibitors TCS PIM-1 4a
Molecular Weight 273.23
Purity >98

Selective, ATP-competitive Pim kinase inhibitor (IC50 values are 24 and 100nM for Pim-1 and Pim-2 respectively). Displays selectivity over a panel of ∽50 other kinases tested. Exhibits cytotoxicity in PC3 prostate carcinoma cells in vitro (IC50 = 17μM).

  • Chemical Name: (5Z)-5-[[3-(Trifluoromethyl)phenyl]methylene]-2,4-thiazolidinedione
  • Formula: C11H6F3NO2S
  • CAS Number: 438190-29-5
  • Solubility: Soluble to 100mM in DMSO and to 100mM in ethanol
  • Purity: >98