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Tocris™ SR 48692

Selective non-peptide NTS1 antagonist

$320.76 - $1,323.85

Specifications

Product Type SR 48692
Inhibitors SR 48692
Molecular Weight 587.07
Purity >98
View More Specs

Disclaimers:

For Research Use Only



Products ${productFamilyLength}
Catalog Number Mfr. No. Quantity Price Quantity  
Catalog Number Mfr. No. Quantity Price Quantity  
372150R Tocris™
RDS372150
50mg Each for $1,323.85
372110R Tocris™
RDS372110
10mg Each for $320.76
Specifications

Description

Neurotensin antagonist; selective for NTS1 over NTS2 (apparent affinity, Ke, is 36nM for NTS1). Competitively inhibits binding of [125I]-neurotensin to HT29 and N1E115 cell membranes (IC50 values are 15.3 and 20.4nM respectively). Orally bioavailable.
  • Chemical Name: 2-[[[1-(7-Chloro-4-quinolinyl)-5-(2,6-dimethoxyphenyl)-1H-pyrazol-3-yl]carbonyl]amino]-tricyclo[3.3.1.13,7]decane-2-carboxylic acid
  • Formula: C32H31ClN4O5
  • CAS Number: 146362-70-1
  • Solubility: Soluble to 20mM in DMSO
  • Purity: >98
Description & Specifications

Specifications

SR 48692
SR 48692
587.07
>98