Please login to your online account to display your discounted pricing

Tocris™ LU AA33810

Potent NPY Y5 receptor antagonist

$199.20 - $841.81

Specifications

Product Type LU AA33810
Inhibitors LU AA33810
Molecular Weight 423.62
Purity >98
View More Specs

 Disclaimers

For Research Use Only

Products
Catalog Number Mfr. No. Quantity Price Quantity    

356210R

 
tocris™
3562/10
10mg Each for $199.20

356250R

 
tocris™
3562/50
50mg Each for $841.81
Description & Specifications

Specifications

Product Type LU AA33810
Inhibitors LU AA33810
Molecular Weight 423.62
Purity >98

Potent neuropeptide Y (NPY) Y5 receptor antagonist (Ki = 1.5nM in vitro). Displays ≥ 3300-fold affinity for Y5 over Y1, Y2 and Y4 receptors. Also binds human 5-HT2B and 5-HT1A receptors (Ki values are 247 and 478nM respectively). Exerts anxiolytic- and antidepressant-like effects in rat models of stress sensitivity.

  • Chemical Name: N-[[trans-4-[(4,5-Dihydro[1]benzothiepino[5,4-d]thiazol-2-yl)amino]cyclohexyl]methyl]methanesulfonamide
  • Formula: C19H25N3O2S3
  • CAS Number: 304008-29-5
  • Solubility: Soluble to 100mM in DMSO
  • Purity: >98