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Tocris™ FR 139317

Highly potent, selective ETA antagonist

Manufacturer:  Tocris™ 121010

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Catalog No. 121010


 

Disclaimers:

For Research Use Only


Specifications

Description

Inhibitor, Enzyme; Tocris; FR 139317; Highly potent, selective ETA antagonist; Molecular wt: 604.75; CAS Number: 142375-60-8; Formula: C33H44N6O5; Purity:>99; 10mg

A highly potent and selective ETA endothelin receptor antagonist (Ki values are 1nM and 7.3μM at ETA and ETB subtypes respectively). Active in vivo.
  • Chemical Name: N-[N-[N-[(Hexahydro-1H-azepin-1-yl)carbonyl]-L-leucyl]-1-methyl-D-tryptophyl]-3-(2-pyridinyl)-D-alanine
  • Formula: C33H44N6O5
  • CAS Number: 142375-60-8
  • Solubility: Soluble to 100mM in 1eq. HCl and to 100mM in DMSO
  • Purity: >99
Description & Specifications

Specifications

FR 139317
>99
10mg
FR 139317
604.75