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Tocris™ CID 16020046

Selective GPR55 antagonist

$250.62 - $1,052.58

Specifications

Product Type CID 16020046
Inhibitors CID 16020046
Molecular Weight 425.44
Purity >99
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 Disclaimers

For Research Use Only

Products
Catalog Number Mfr. No. Quantity Price Quantity    

495910R

 
tocris™
4959/10
10mg Each for $250.62

495950R

 
tocris™
4959/50
50mg Each for $1,052.58
Description & Specifications

Specifications

Product Type CID 16020046
Inhibitors CID 16020046
Molecular Weight 425.44
Purity >99

Selective GPR55 antagonist. Inhibits LPI-induced Ca2+ signaling (IC50 = 0.21μM in HEK-GPR55 cells), ERK1/2 phosphorylation and GPR55-mediated transcription factor activation. Displays weak inhibition of acetylcholinesterase,μ-opioid receptor, KCNH2 and hERG. Decreases LPI-induced GPR55 internalization. Reduces experimental intestinal inflammation in mice.

  • Chemical Name: 4-[4,6-Dihydro-4-(3-hydroxyphenyl)-3-(4-methylphenyl)-6-oxopyrrolo[3,4-c]pyrazol-5(1H)-yl]benzoic acid
  • Formula: C25H19N3O4
  • CAS Number: 834903-43-4
  • Solubility: Soluble to 100mM in DMSO
  • Purity: >99